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binds convincingly within the ATP-binding site of Pim-1 suggesting an ATP-competitive inhibitory mechanism
CN1[C@@H]2C[C@@H](O)C[C@H]1[C@@H]1O[C@H]21
active-site directed and substrate competitive AKR1C1 inhibitor (Ki = 4 nM) with moderate to excellent selectivity over AKR1C2
InChi: InChI=1S/C25H34F2O5/c1-18(2)32-24(30)13-9-4-3-8-12-20-21(23(29)16-22(20)28)14-15-25(26
Liproxstatin-1 (10 mg/kg
Telotristat 845 binds convincingly within the ATP-bindingTelotristat, also known as LP 778902, is the acid form of Telotristat ethyl, and the active metabolite of LX1606 (Telotristat etiprate), which is an orally bioavailable, small molecule, tryptophan hydroxylase (TPH) inhibitor and serotonin synthesis inhibitor with potential antiserotonergic activity. Blocking peripheral serotonin synthesis by telotristat reduces severity of both chemical and infection induced intestinal inflammation. Product